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Argentine Researchers Validate RAC1 Blockade to Protect the Liver in Fulminant Hepatitis

An oncology‑derived compound cut injury markers in animals and human liver explants, and the program now aims for regulated toxicology and clinical testing.

Overview

  • The molecule 1D-142, originally developed for cancer, produced 40%–60% reductions in ALT and AST and lowered inflammation, necrosis and reactive oxygen species across three animal models.
  • In ex vivo human liver explants from acute liver failure patients, treatment decreased necrosis and inflammatory signals, with no toxicity detected in healthy liver samples.
  • The work was led by the Laboratorio de Hepatología Experimental y Terapia Génica (Universidad Austral/CONICET) with contributions from INTI and biotech partner Spectrum.
  • The study has been accepted by Journal of Hepatology Reports and forms part of Bárbara Bueloni’s doctoral research under Guillermo Mazzolini and Juan Bayo.
  • An international PCT patent is pending, and investigators report a newly identified molecule with potentially greater potency while emphasizing the findings remain preclinical and funding and trials are needed.